「receptors」の共起表現一覧(2語左で並び替え)
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The type A GABA | receptors are pentameric chloride channels assembled f |
binding and signaling through a TrkC-related | receptors called TrkB. |
It can act on | receptors at pre-ganglionic sites in both the sympathe |
es can act in numerous ways, often acting as | receptors or ligands (the molecule that activates a re |
cell contact, ion conductance, and acting as | receptors. |
of flunisolide is to activate glucocorticoid | receptors. |
elatively wide gap (>20 µm) to activate 5-HT | receptors located on the dendrites, cell bodies and pr |
ere are 11 growth factors that activate ErbB | receptors. |
Like capsaicin, capsinoids activate TRPV1 | receptors, although they are not hot in the mouth. |
both capsaicin and capsinoids activate TRPV1 | receptors in the same manner. |
promotion sites by ligand activated nuclear | receptors. |
Activated I1-imidazoline | receptors trigger the hydrolysis of phosphatidylcholin |
gonist is a compound that activates dopamine | receptors in the absence of dopamine. |
IP3 enters the cytoplasm and activates IP3 | receptors on the smooth endoplasmic reticulum (ER), wh |
rmone cortisol that activates glucocorticoid | receptors. |
ediated effects but also activates adenosine | receptors, often with opposing (patho-) physiological |
ns that serotonin has when it activates 5-HT | receptors. |
uronal signaling molecule by activating NMDA | receptors in the brain. |
al selectivity by strongly activating 5-HT1A | receptors in the prefrontal cortex while having little |
By activating 5-HT2C | receptors, vabicaserin inhibits dopamine release in th |
periments using constitutively active BMPR1B | receptors. |
ceptor and reverses constitutive activity of | receptors. |
ts there are yet more additional cannabinoid | receptors. |
Adenosine A3 | receptors are G protein-coupled receptors that are inv |
anchored cytokines, cell adhesion molecules, | receptors, ligands, and enzymes. |
Adopted orphan | receptors in the nuclear receptor group include the fa |
localizes with intracellular adrenal steroid | receptors and converts cortisol (an active mineralcort |
dy produces antibodies against acetylcholine | receptors, and thus inhibits signal transmission acros |
The renal effects allow the | receptors to change the mean pressure in the system in |
he rat parotid gland and at alpha adrenergic | receptors. |
partial agonist action at Alpha-2 adrenergic | receptors, and TDIQ has been suggested as a possible d |
ular domain of the protein which is also the | receptors G protein coupling domain.Therefore editing |
tain CCKBR (which respond to gastrin) and M3 | receptors (which respond to Ach). |
cannabinoid agonist at both the CB1 and CB2 | receptors. |
rect or indirect activation of CB2 and TRPV1 | receptors, and induction of oxidative stress, all cont |
as a low affinity for AMPA, kainate and NMDA | receptors. |
y over the closely related 5-HT2A and 5-HT2B | receptors. |
onsidered a full agonist at both CB1 and CB2 | receptors and has Ki values of 0.58nM and 0.68nM respe |
mary actions of steroid hormones and nuclear | receptors. |
energic, α2-adrenergic, β-adrenergic, and D2 | receptors. |
nates are innervated by pain and temperature | receptors, via the trigeminal nerve (or, the fifth cra |
pe I (I and IB) and two type II (II and IIB) | receptors. |
a selective antagonist at dopamine D2 and D3 | receptors. |
It has high affinity for both CB1 and CB2 | receptors, with Ki values of 1.5nM at CB1 and 0.32nM a |
ive in synthesizing shape- and ion-selective | receptors, and throughout the 1980s research in the ar |
selective agonist for the 5-HT2A and 5-HT2C | receptors, but unlike the corresponding benzocyclobute |
r binding affinity for the 5-HT1A and 5-HT2A | receptors, but is less potent in producing drug-approp |
eceptor full agonist at both the CB1 and CB2 | receptors. |
MG-3 is a potent agonist at both CB1 and CB2 | receptors with a Ki of 0.32nM at CB1 and 0.52nM at CB2 |
, the macrophage expresses more CD40 and TNF | receptors on its surface which helps increase the leve |
idence for receptor overexpression and spare | receptors suggests that the calculation of the net cha |
cardioselectivity and blocks both β1 and β2 | receptors. |
as fairly high affinity for both CB1 and CB2 | receptors, with Ki values of 2.91nM at CB1 and 4.24nM |
through a site separate from the CB1 and CB2 | receptors, which responds to abnormal cannabidiol, O-1 |
ved to work by blockading dopamine D1 and D2 | receptors in the mesocortical and mesolimbic pathways, |
ctive full agonist at the dopamine D1 and D5 | receptors. |
acts as an agonist at the 5-HT1A and 5-HT1B | receptors and as an antagonist at the 5-HT2C receptor. |
signaling pathways, coregulators and nuclear | receptors at a promoter showing local nucleosomal cond |
receptor, a weak agonist at both CB1 and CB2 | receptors, and an inhibitor of anandamide reuptake. |
y over the closely related 5-HT1D and 5-HT1A | receptors. |
has some affinity for the 5-HT2A and 5-HT2C | receptors, though it is unlikely that these properties |
cannabinoid agonist at both the CB1 and CB2 | receptors, but with moderate selectivity for CB2, havi |
For example, P2X1 and P2X3 | receptors desensitize rapidly (a few hundred milliseco |
al class that acts on serotonin and dopamine | receptors. |
e I ( I and IB) and two type II (II and IIB) | receptors. |
o other areas of the brain, and somatostatin | receptors are expressed at many different sites in the |
BN acts as a weak agonist of the CB1 and CB2 | receptors, with lower affinity in comparison to THC. |
be an antagonist at the GABAA and GABAA-rho | receptors. |
or adrenergic, histaminergic, and muscarinic | receptors. |
y over the closely related 5-HT2A and 5-HT2C | receptors. |
s the neurons by activating AMPA and kainate | receptors, causing an influx of calcium. |
cannabinoid agonist at both the CB1 and CB2 | receptors. |
albicans as virulence factors and toll-like | receptors as relevant mediators of the inflammatory ho |
ately equal affinity at both the CB1 and CB2 | receptors, having a Ki of 8.0nM at CB1 and 7.0nM at CB |
is a potent agonist at both the CB1 and CB2 | receptors, with a binding affinity of 0.1nM at CB1 and |
Chemokines and their | receptors are important for the migration of various c |
cannabinoid agonist at both the CB1 and CB2 | receptors. |
x selectivity over the related Y1, Y2 and Y4 | receptors. |
s of beta receptor, designated β1, β2 and β3 | receptors. |
Several ion channels and neurotransmitters | receptors pre-mRNa are substrates for ADARs. |
Chemokines and their | receptors are key regulators of the thymocytes migrati |
s in the skin also express NMDA and non-NMDA | receptors. |
The D1 and D5 | receptors are members of the D1-like family of dopamin |
ptor antagonist, antagonizing A1, A2, and A3 | receptors almost equally, which explains many of its c |
Type I and II | receptors form a stable complex after ligand binding, |
has shown that the nicotinic and muscarinic | receptors belong to distinct protein superfamilies. |
itionally affinity for the 5-HT2A and 5-HT2C | receptors. |
It acts on D1 and α | receptors as a agonist. |
the estrogen, androgen and mineralocorticoid | receptors. |
ylcholine, GABAA, GABAA-ρ, glycine and 5-HT3 | receptors that are composed of five protein subunits w |
s found to be an agonist at both CB1 and CB2 | receptors. |
a ligand for various serotonin and dopamine | receptors. |
t has moderate affinity for both CB1 and CB2 | receptors, with Ki values of 8.36nM at CB1 and 7.95nM |
tive for the β1-adrenergic and β2-adrenergic | receptors. |
cterising the active site of the CB1 and CB2 | receptors. |
rongest actions are at the 5-HT2B and 5-HT2C | receptors and its discriminative cue is mediated prima |
interact with muscarinic-2 and muscarinic-4 | receptors to inhibit neurally released acetylcholine. |
binds to the glucocorticoid and progesterone | receptors and therefore blocks the activity of the end |
rons may interact with alpha-2A and alpha-2C | receptors to inhibit neurally released norepinephrine. |
utoreceptor similar to the 5-HT1B and 5-HT1D | receptors. |
It stimulates dopaminergic and serotonergic | receptors and blocks alpha-adrenoreceptors. |
tant for neutrophils acting at BLT1 and BLT2 | receptors on the plasma membrane of these cells. |
entan), which affect both endothelin A and B | receptors. |
Other neurokinin subtypes and neurokinin | receptors that interact with SP have also been reporte |
sm is facilitated by D2/D3, nACh, and 5-HT2A | receptors. |
and has modest affinity for both CB1 and CB2 | receptors, with Ki values of 48.3nM at CB1 and 45.5nM |
It acts as an agonist at the 5HT2A and 5HT2C | receptors. |
with the exception of the 5-HT2A and 5-HT2C | receptors where it acts as a partial agonist. |
cannabinoid agonist at both the CB1 and CB2 | receptors. |
racts centrally with dopamine and adrenergic | receptors. |
Warm and cold | receptors play a part in sensing innocuous environment |
mitragynine acts on the mu- and delta-opiate | receptors. |
hibitor and agonist at the 5-HT2A and 5-HT2C | receptors. |
lectivity over the related 5-HT2B and 5-HT2C | receptors. |
ulation, molecular endocrinology and steroid | receptors and transcriptional coactivators. |
cannabinoid agonist at both the CB1 and CB2 | receptors, with Ki values of 0.46nM at CB1 and 0.69nM |
that the differences between GABAС and GABAA | receptors are large enough to justify maintaining the |
lso partial agonist of µ-opioid and δ-opioid | receptors, and competitive antagonist of ϰ-opioid rece |
high affinity for the dopamine D2, D3 and D4 | receptors, as well as serotonin 5-HT1A and 5-HT2A/C re |
ist with high affinity to the D2, D3, and D4 | receptors, and with moderate affinity for the 5-HT2 re |
y over the closely related 5-HT1D and 5-HT1A | receptors. |
, and cytoskeletal organization and syndecan | receptors are required for internalization of the HIV- |
e, suggesting a role for the 5-HT6 and 5-HT7 | receptors in regulation of the hearing system. |
the antigen receptor (TCR) and costimulatory | receptors (CD28 and ICOS) are thought to be main recep |
The D1 and D5 | receptors have a high degree of structural homology an |
selective for Y4 over the related Y1 and Y5 | receptors, as the first non-peptide Y4 antagonist deve |
Unlike the H1 and H2 | receptors which have primarily peripheral actions, but |
lectivity over the related 5-HT2A and 5-HT2C | receptors. |
HT2C), 5-HT6, 5-HT7, α1-adrenergic, and NMDA | receptors, and as agonists at the sigma receptors (σ1 |
activated so that the actions of the δ and κ | receptors can be studied separately, in contrast to be |
d efficacious agonist at the M1 and δ-opioid | receptors, unlike clozapine as well. |
s, including stimulation of alpha and beta-1 | receptors and inhibition of noradrenaline and tyramine |
oximately equal affinity for the CB1 and CB2 | receptors, with a Ki of 6.6nM at CB1 and 6.9nM at CB2. |
, the ATP sensitivity of P2X1, P2X3 and P2X4 | receptors is attenuated when the extracellular pH<7, w |
hannels including the GABAA, NMDA, and sigma | receptors. |
y over the closely related 5-HT2A and 5-HT2C | receptors and other receptor targets. |
t as non-selective antagonists at A1 and A2A | receptors in both heart and brain and so have the oppo |
ptor alpha, a subunit shared by IL13 and IL4 | receptors. |
antagonist at various serotonin and dopamine | receptors. |
0 mg/day due to its ability to antagonise H3 | receptors and thus increase the release of serotonin a |
uscle rather than by antagonizing muscarinic | receptors. |
M, and no significant affinity for any other | receptors tested. |
eptor" family of apoptosis-inducing cellular | receptors. |
of its potency, because the appropriate CB1 | receptors are not located in brain areas reponsible fo |
Several of these are Integrin | receptors. |
There are numerous | receptors that now known to use intracellular kinases |
In biochemistry, there are decoy | receptors, decoy substrates and decoy RNA. |
d to a discovery that there are cell-surface | receptors that are stimulated by hormones and neurotra |
n potential formation, there are not as many | receptors for GABA to bind to - meaning that sympathet |
ts like osteoprotegerin as both act as decoy | receptors for osteoblastic RANKL. |
stranded DNA) molecules which act as surface | receptors. |
of deep burn there will be no pain as these | receptors will be burned off. |
As IP3 | receptors have sparse or little distribution throughou |
clear receptor family such as glucocorticoid | receptors. |
antiadhesive agents, and second as adhesion | receptors. |
eins that appear to function as cell-surface | receptors for Wnts. |
PKC family members also serve as major | receptors for phorbol esters, a class of tumor promote |
CD16 has been identified as Fc | receptors FcγRIIIa and FcγRIIIb. |
ked to the D3 activity of pramipexole, as D3 | receptors are heavily expressed in brain regions invol |
egral proteins that function as cell-surface | receptors for Wnts called serpentine receptors. |
Hence NCOA2 assists nuclear | receptors in the upregulation of DNA expression. |
Muscles and associated sensory | receptors are innvervated by type I and II sensory fib |
rimary tumor mass, and if HA associates with | receptors such as CD44, the activation of Rho GTPases |
ed to THC, which is a partial agonist at CB1 | receptors, JWH-018 (and many of its analogues) are ful |
lecule to continuously bind and unbind at β2 | receptors in the smooth muscle in the lungs. |
acts as a nonselective full agonist at GABAA | receptors. |
selective, mixed agonist-antagonist at GABAA | receptors, which acts as a partial agonist at the α2 a |
culline, ROD-188 acts as an agonist at GABAA | receptors, being a positive allosteric modulator actin |
acts as a partial agonist at benzodiazepine | receptors. |
ative drug which acts as an agonist at GABAA | receptors, specifically acting as a positive allosteri |
a subtype-selective partial agonist at GABAA | receptors, and was developed by Pfizer as a potential |
as, , had a direct action at pharmacological | receptors and thereby acting as a neurotransmitter was |
shown to possess some activity at serotonin | receptors. |
n the mammalian brain where it acts at GABAA | receptors, which are ligand-gated chloride channels. |
the mammalian brain where it acts at GABA-A | receptors, which are ligand-gated chloride channels. |
Meclozine is an antagonist at H1 | receptors. |
cts as a partial agonist/antagonist at these | receptors. |
t acts as an inverse agonist at melanocortin | receptors, specifically, MC1. |
ts also commonly have action at α-adrenergic | receptors and/or 5-HT receptors. |
in the mammalian brain where it acts at GABA | receptors, which are ligand-gated chloride channels. |
e action of aldosterone at mineralocorticoid | receptors. |
te, some of which also act at benzodiazepine | receptors. |
the estrogenic potency of coumestrol at both | receptors is much less than that of 17β-estradiol. |
a subtype-selective partial agonist at GABAA | receptors, with highest affinity for the α3 subtype, b |
subtype, and little or no affinity at other | receptors. |
4 is a nonselective partial agonist at GABAA | receptors. |
nvulsant shown to act as an agonist at GABAA | receptors. |
the mammalian brain where it acts at GABA-A | receptors, which are ligand-gated chloride channels. |
The weak agonist activity of pergolide at D1 | receptors somewhat alters its clinical and side effect |
It is a partial agonist at CB1 | receptors, with a Ki of 87nM, making it roughly half t |
esearch which acts as an antagonist at GABAB | receptors. |
t but non-selective partial agonist at GABAA | receptors, although with little efficacy at the α1 sub |
Semorphone is a partial agonist at μ-opioid | receptors. |
ion of 2-heptanone as a pheromone at odorant | receptors in mice has been investigated. |
It is a partial agonist acting at GABAA | receptors in the brain. |
211, is a mixed agonist-antagonist at opioid | receptors with a similar pharmacological profile to pe |
phic factor (BDNF), glutamate acting at NMDA | receptors, dopamine through activation of the D1 recep |
subtype, with little or no affinity at other | receptors. |
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