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出典:『Wikipedia』 (2011/02/12 21:22 UTC 版)

英語による解説

引用

AM-855 is an analgesic drug which is a cannabinoid agonist. It is a derivative of Δ⁸Tetrahydrocannabinol with a conformationally restricted side chain which has been bound into a fourth ring fused to the aromatic A-ring of the cannabinoid skeleton. AM-855 is an agonist at both CB1 and CB2 with moderate selectivity for CB₁, with a Ki of 22.3nM at CB₁ and 58.6nM at CB₂.