出典:Wiktionary
出典:『Wiktionary』 (2010/07/01 16:17 UTC 版)
vanoxerine (uncountable)
出典:Wikipedia
出典:『Wikipedia』 (2011/06/22 11:43 UTC 版)
Vanoxerine (GBR-12909) is a piperazine derivative which is a potent and selective DRI. GBR-12909 binds to the target site on the DAT ~ 500 times more strongly than cocaine, but simultaneously inhibits the release of dopamine. This combined effect only slightly elevates dopamine levels, giving vanoxerine only mild stimulant effects.