「receptors」の共起表現一覧(1語右で並び替え)
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to PPARs (peroxisome proliferator-activated | receptors), a group of receptor molecules inside the c |
nably selective antagonist for the adenosine | receptors A1 and A2A, having a Ki of 3.3nM at A2A and |
ntagonism of presynaptic inhibitory dopamine | receptors accounting for some antidepressant activity |
M2 muscarinic | receptors act via a Gi type receptor, which causes a d |
ective mixed agonist-antagonist for dopamine | receptors, acting as a weak partial agonist at the D3 |
onist at α4β2 neural nicotinic acetylcholine | receptors, acting as an agonist at (α4)2(β2)3 pentamer |
Tyrosine kinase growth factor | receptors activate mitogen-activated protein kinases w |
1 over D5 with negligible affinity for other | receptors; acts as an antagonist at D1 but as an agoni |
There are three type I Activin | receptors: ACVR1, ACVR1B, and ACVR1C. |
inding domain of HNF4, as with other nuclear | receptors, adopts a canonical alpha helical sandwich f |
The | receptors affect the downstream target AMP kinase, an |
Retrovirus | receptors allow infection of human and murine cells by |
s along with the five different somatostatin | receptors allows somatostatin to possess a large range |
ptor antagonist, antagonizing A1, A2, and A3 | receptors almost equally, which explains many of its c |
Increased firing from the stretch | receptors also increases production of pulmonary surfa |
Receptors also have varying affinities for odorant mol | |
However, metabotropic | receptors also remain open from seconds to minutes (Ka |
ally show no affinity for the most important | receptors, although modulation of most important centr |
nd anxiolytic effects is by modulating GABAA | receptors, although suriclone is more subtype-selectiv |
ide antagonist selective for the neurotensin | receptors, although not selective between subtypes. |
ts anxiolytic effects is by modulating GABAA | receptors, although ocinaplon is more subtype-selectiv |
t but non-selective partial agonist at GABAA | receptors, although with little efficacy at the α1 sub |
Like capsaicin, capsinoids activate TRPV1 | receptors, although they are not hot in the mouth. |
as a partial agonist at GABAA benzodiazepine | receptors, although pazinaclone is more subtype-select |
tragynine itself acts primarily via μ-opioid | receptors, although its oxidation product mitragynine- |
moniae that seemed to involve an exchange of | receptors among diverse bacteria either grown together |
teins (RAMPs), forming the multimeric amylin | receptors AMY1 (CT + RAMP1), AMY2 (CT + RAMP2), and AM |
with around 70x selectivity for OX1 over OX2 | receptors, and improved oral bioavailability compared |
h show little or no affinity to other opioid | receptors and so allow ORL-1 mediated responses to be |
rect or indirect activation of CB2 and TRPV1 | receptors, and induction of oxidative stress, all cont |
onsidered a full agonist at both CB1 and CB2 | receptors and has Ki values of 0.58nM and 0.68nM respe |
ive in synthesizing shape- and ion-selective | receptors, and throughout the 1980s research in the ar |
ntaining a striped expression pattern of Eph | receptors and their ligands, which is vital to proper |
properties (potentiation of interferon gamma | receptors and production), DIM is also under investiga |
a subtype-selective partial agonist at GABAA | receptors, and was developed by Pfizer as a potential |
It has been found to inhibit histamine H1 | receptors and platelet aggregation, and acts as an opi |
as, , had a direct action at pharmacological | receptors and thereby acting as a neurotransmitter was |
the fact that it has high affinity for both | receptors and stimulates the D5-linked PLC/PI second m |
rovides a liver with normally functional LDL | receptors, and leads to rapid improvement of the chole |
acts as an agonist at the 5-HT1A and 5-HT1B | receptors and as an antagonist at the 5-HT2C receptor. |
receptor, a weak agonist at both CB1 and CB2 | receptors, and an inhibitor of anandamide reuptake. |
partial agonist action at Alpha-2 adrenergic | receptors, and TDIQ has been suggested as a possible d |
(dPTX) is most effective to block glutamate | receptors and especially those quisqualate-sensitive, |
t adenylate cyclases may couple to olfactory | receptors and that there may be multiple receptor-medi |
ive for the ORL-1 receptor over other opioid | receptors, and its effects in animals include preventi |
cid binding Ig-like lectins are cell surface | receptors and members of the immunoglobulin superfamil |
eline, an agonist on Ganglion type nicotinic | receptors and also affects sensory nerve terminals |
ation that inhibits muscarinic acetylcholine | receptors and thus the parasympathetic nervous system. |
pericine has been shown to bind to mu opioid | receptors, and has an IC50 of 0.6μmol, around 6x more |
specialize in binding to erythrocyte surface | receptors and facilitating erythrocyte entry. |
ptor β is a member of the family of estrogen | receptors and the superfamily of nuclear receptor tran |
th either GRIK4 or GRIK5 to form heteromeric | receptors and acts as an excitatory neurotransmitter a |
rations actually prevent dimerization of the | receptors and prevent signalling. |
d imidazoline binding sites, and blocks NMDA | receptors and other cation ligand-gated channels. |
Quisqualic acid is an agonist for both AMPA | receptors and group I metabotropic glutamate receptors |
of agonists acting through G protein-coupled | receptors and receptor tyrosine kinases stimulate this |
an agonist at neural nicotinic acetylcholine | receptors and has been researched for use as an analge |
These saturate the | receptors and prevent T cell activation and thus preve |
gerol as a high affinity agonist for alpha-2 | receptors and a medium affinity antagonist at the 5-HT |
The PI3K is activated by G protein-coupled | receptors and tyrosine kinase receptors. |
has been investigated for its effect on AMPA | receptors and researched for potential use in the trea |
ocriptine is a potent agonist at dopamine D2 | receptors and various serotonin receptors. |
It binds to all known somatostatin | receptors, and shares many pharmacological and functio |
Steroid hormone | receptors and related receptors are generally soluble |
mones at Chicago, where he isolated estrogen | receptors and discovered their importance in breast ca |
2-AG can also activate both cannabinoid | receptors and is inactivated by monoacylglycerol lipas |
dy produces antibodies against acetylcholine | receptors, and thus inhibits signal transmission acros |
lacks any significant affinity for adenosine | receptors and does not produce stimulant effects. |
eficiency is a defect in the body's cytokine | receptors and their signaling. |
ese include the Toll family of innate immune | receptors and the receptor for IL-18. |
benzodiazepines, lacking affinity for GABAA | receptors and instead acting as a cholecystokinin anta |
Various Eph | receptors and ephrins are expressed in these regions, |
neurotransmitters which interact with nerve | receptors and smooth muscle cells. |
rongest actions are at the 5-HT2B and 5-HT2C | receptors and its discriminative cue is mediated prima |
ving amongst others an interaction between δ | receptors and mitochondrial K(ATP) channels. |
The venom blocks octopamine | receptors and the cockroach fails to show normal escap |
antagonist action at nicotinic acetylcholine | receptors, and it has also been shown to reduce the co |
The diverse feature of the chemotaxis | receptors and ligands provides the possibility to sele |
binds to the glucocorticoid and progesterone | receptors and therefore blocks the activity of the end |
It stimulates dopaminergic and serotonergic | receptors and blocks alpha-adrenoreceptors. |
e derived from A domains of various membrane | receptors and have a rigid structure, stabilised by di |
s down-regulation of Ca2+ -impermeable GluR2 | receptors and inhibits calpain, a Ca2+ -activated prot |
macromolecular systems such as ion channels, | receptors, and protein kinases. |
nded research consortium focussed on nuclear | receptors and nuclear receptor coregulators. |
s is the influx of calcium through the NMDAR | receptors and the resultant activation of Ca2+/calmodu |
re mediated through muscarinic acetylcholine | receptors and can be prevented by prior administration |
ce, Senomyx has identified hundreds of taste | receptors and currently owns 113 patents on their disc |
e, but it does not act at the classic opioid | receptors and its actions are not antagonized by the o |
of a variety of ion channels, including NMDA | receptors and AMPA receptors. |
This can bind to Interleukin-2 | receptors and introduce the diphtheria toxin into cell |
ergic, adrenergic, muscarinic or cannabinoid | receptors and does not block potassium or calcium curr |
ulation, molecular endocrinology and steroid | receptors and transcriptional coactivators. |
lso partial agonist of µ-opioid and δ-opioid | receptors, and competitive antagonist of ϰ-opioid rece |
ist with high affinity to the D2, D3, and D4 | receptors, and with moderate affinity for the 5-HT2 re |
negligible affinity for the 5-HT1A or 5-HT2C | receptors, and over 400-fold lower affinity for the D2 |
0 mg/day due to its ability to antagonise H3 | receptors and thus increase the release of serotonin a |
ule that interacts with various cell surface | receptors and mediates cell apoptotic signals. |
Title: Interactions of Eph-related | receptors and ligands confer rostrocaudal pattern to t |
a selective radioligand for the cannabinoid | receptors and has been used as its 131I derivative for |
It is a partial agonist of benzodiazepine | receptors and has been shown to possess both anxiolyti |
st likely caused by activity at kappa opioid | receptors and sigma receptors. |
It belongs to the type I cytokine | receptors, and has been shown to form a heterodimeric |
gonist-antagonist at nicotinic acetylcholine | receptors and an antagonist at μ-opioid receptors. |
-Bungarotoxin blocks nicotinic acetylcholine | receptors and has been used to isolate and study them; |
localizes with intracellular adrenal steroid | receptors and converts cortisol (an active mineralcort |
HT2C), 5-HT6, 5-HT7, α1-adrenergic, and NMDA | receptors, and as agonists at the sigma receptors (σ1 |
it possesses intrinsic activity at the D2/D3 | receptors, and acts as a weak partial agonist at these |
modes of action such as through histamine H3 | receptors and glutamate. |
s, including stimulation of alpha and beta-1 | receptors and inhibition of noradrenaline and tyramine |
various experiments to sever Westlake's pain | receptors and enhance his strength to superhuman level |
eraction with G-protein-coupled somatostatin | receptors and inhibition of the release of numerous se |
Palifermin binds to epithelial cell-surface | receptors and stimulates epithelial cell proliferation |
bitter taste work through G protein-coupled | receptors, and the savory sensation is activated by gl |
s as a positive allosteric modulator of AMPA | receptors, and has nootropic effects in animal studies |
y over the closely related 5-HT2A and 5-HT2C | receptors and other receptor targets. |
s act through intracellular (mostly nuclear) | receptors and, thus, are considered to be intracrines. |
ts also commonly have action at α-adrenergic | receptors and/or 5-HT receptors. |
The C-terminus of CB2 | receptors appears to play a critical role in the regul |
The M2 muscarinic | receptors are located in the heart, where they act to |
Typically type II cytokine | receptors are hetrodimers or multimers with a high and |
These | receptors are related predominantly by sequence simila |
Complement | receptors are responsible for detecting pathogens by m |
Muscarinic | receptors are found in both the central nervous system |
For example, 5-HT1E | receptors are abundant in the hippocampus but are not |
Most frizzled | receptors are coupled to the beta-catenin canonical si |
ding the interaction of losigamone with GABA | receptors are inconsistent: it increases GABA-induced |
It is now known that S1P | receptors are members of the Lysophospholipid receptor |
r antidepressant on various transporters and | receptors are summarized below. |
Chemotaxis | receptors are expressed in the surface membrane with d |
The CB2 | receptors are found primarily on microglia(the immune |
GABAB | receptors are involved in behavioral actions of ethano |
Cytokine | receptors are receptors that bind cytokines. |
Muscarinic | receptors are metabotropic, and affect neurons over a |
These methyl-accepting chemotaxis | receptors are one of the first components in the senso |
TGFβ | receptors are single pass serine/threonine kinase rece |
o other areas of the brain, and somatostatin | receptors are expressed at many different sites in the |
Imidazoline | receptors are receptors for clonidine and other imidaz |
The angiopoietin | receptors are receptors that bind angiopoietin. |
Ion channel linked | receptors are cell membrane bound receptors. |
CB2 | receptors are also found throughout the gastrointestin |
These | receptors are heteromeric protein complexes with multi |
The two main types of glutamate | receptors are ionotropic receptors and metabotropic re |
These olfactory | receptors are membrane proteins of bipolar olfactory r |
The ligands of these | receptors are members of the TGF beta superfamily. |
The asialoglycoprotein | receptors are lectins which bind asialoglycoprotein, g |
Several other LIR subfamily B | receptors are expressed on immune cells where they bin |
β3-adrenergic | receptors are located in fat cells. |
The type A GABA | receptors are pentameric chloride channels assembled f |
β2-adrenergic | receptors are located mainly in the lungs, gastrointes |
These | receptors are found in the central and peripheral auto |
Eph | receptors are components of cell signalling pathways i |
Peptide hormone | receptors are often transmembrane proteins. |
Galanin | receptors are seven-transmembrane proteins shown to ac |
N-methyl-D-aspartate (NMDA) | receptors are a class of ionotropic glutamate receptor |
Retinoid | receptors are nuclear receptors (a class of proteins) |
These | receptors are also closely related to the activin rece |
Chemokines and their | receptors are important for the migration of various c |
β1-adrenergic | receptors are located mainly in the heart and in the k |
These | receptors are all transmembrane proteins, composed of |
Chemokines and their | receptors are key regulators of the thymocytes migrati |
most important functions of thyroid hormone | receptors are regulation of metabolism and heart rate. |
of its potency, because the appropriate CB1 | receptors are not located in brain areas reponsible fo |
Examples of such tonic | receptors are pain receptors, joint capsule, and muscl |
Glutamate | receptors are (as mentioned above) also expressed in p |
Sigma | receptors are affected by cocaine, as cocaine function |
The D1 and D5 | receptors are members of the D1-like family of dopamin |
These | receptors are similar to type I cytokine receptors exc |
Type I | receptors are essential for signaling, and type II rec |
Type I | receptors are essential for signaling; and type II rec |
These | receptors are predominately expressed in cells of the |
Expression of the | receptors are correlated with insulin levels, as well |
Examples of orphan | receptors are found in the G protein-coupled receptor |
V1 | receptors are found in various sites around the body. |
alpha7-containing | receptors are known to improve prepulse inhibition, pr |
G protein-coupled | receptors are composed of seven membrane-spanning alph |
Most older compounds acting on adenosine | receptors are nonselective, with the endogenous agonis |
The three | receptors are dominated by three rhodopsin-like pigmen |
ked to the D3 activity of pramipexole, as D3 | receptors are heavily expressed in brain regions invol |
Pulmonary stretch | receptors are mechanoreceptors found in the lungs. |
Type II | receptors are considered to be constitutively active k |
Signalling outputs from these | receptors are influenced both by the binding of the ch |
tagonists (BQ-788) which affect endothelin B | receptors are used in research but have not yet reache |
The LDL | receptors are minimally functional, if at all. |
Ion-channel-linked | receptors are also called ligand-gated channels. |
Soluble cytokine | receptors are extremely common regulators of cytokine |
Glucagon | receptors are mainly expressed in liver and in kidney |
5HT-3 | receptors are responsible for causing many things from |
Since the antigen | receptors are typically composed of two variable domai |
Merkel | receptors are also located in the mammary glands. |
Most enzyme-linked | receptors are of this type. |
e most active areas of search for ligands to | receptors, are in the field of brain receptors. |
The ligands for these | receptors are free fatty acids (FFAs) and eicosanoids. |
Upon activation, "low-affinity" IL-2 | receptors are replaced by "high-affinity" IL-2 recepto |
netic tree showing how a number of monoamine | receptors are related to each other. |
Some tonic | receptors are permanently active and indicate a backgr |
However since GABAС | receptors are closely related in sequence, structure, |
Neurotrophin ligands of Trk | receptors are processed ligands, meaning that they are |
ErbB | receptors are made up of an extracellular region or ec |
Metabotropic | receptors are G-protein coupled receptors that mediate |
that the differences between GABAС and GABAA | receptors are large enough to justify maintaining the |
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