rti-55とは 意味・読み方・使い方

(–)-2β-Carbomethoxy-3β-(4-iodophenyl)tropane (β-CIT, RTI-55, iometopane) is a phenyltropane-based psychostimulant used in scientific research and with some medical application/s. This drug was first cited in 1991. RTI-55 is a dirty DRI derived from methylecgonidine. RTI-55 is one of the most potent phenyltropane stimulants commercially available, which limits its use in humans, as it might have significant abuse potential if used outside of a strictly controlled medical setting. In contrast to RTI-31 which is predominantly dopaminergic, increasing the size of the covalently bonded halogen from a chlorine to an iodine markedly increases the affinity for the SERT, while retaining mostly all of its DAT blocking activity.